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Chemical name Usage
N2-[(1S)-Ethoxycarbonyl-3-phenylpropyl]-L-alanine Antihypertensives (Enalapril etc.)
1-[(2,3-Dihydro-1,4-benzodioxan-2-yl) carbonyl] piperazine Antihypertensives
(Doxazosin Mesylate etc.)
6,7-Dimethoxy-2-(1-Piperazinyl)-Quinazoline Antihypertensives
(Doxazosin Mesylate etc.)
N-(2-Tetrahydro furoyl) Piperazine Antihypertensives
(Terazosin HCL etc.)
2-Chloromethyl-3,5-dimethyl-4-methoxy pyridine
 hydrochloride
Antiulceratives (Omeprazole etc.)
1-[(2,3-Dichlorophenyl)piperazine hydrochloride Antipsychotics(Aripiprazole etc.)
L (+) Diethyl tartrate  Antiulceratives(Dexlansoprazole etc)
3,4-Dihydroxy-5-nitro benzaldehyde Antiparkinisonians(Entacapone etc)
2-(1H-indol-5-yl)-N-methyl ethane sulfonamide Antimigraines(Naratriptan HCl etc.)
(R)-5-Bromo-3-[(1-methyl-2-pyrrolidinyl)methyl]-1H-indole Antimigraines(Eletriptan HBr etc.)
phenyl vinyl sulfone Antimigraines(Eletriptan HBr etc.)
(R)-(-)-1-Indanamine hydrochloride Antiparkinsonians(Rasagiline Mesylate etc)
(R)-(-)-1-Indanamine Antiparkinsonians(Rasagiline Mesylate etc) 
44-(2-Fluora-4-nitrophenyl)morpholine Antibacterials(Linezolid etc.)
43-fluro-4-morpholinoaniline Antibacterials(Linezolid etc)
4(S)-5-(Aminomethyl)-3-(3-fluoro-4-morpholiniphenyl)oxozolidin-2-one Antibacterials(Linezolid etc)
N-(2-(Benzyloxy)pentan-3-yl)formohydrazide Antifungals(posaconazole etc)
(5R-Cis)-Toluene-4-sulfonicacid-5-(2,4-difluorophenyl)-5-(1H-1,2,4-triazol-1-yl)methyltetrahydrofuran 3-ylmethyl ester Antifungals(posaconazole etc)
2-[(1S,2S)-1-Ethyl-2-benzyloxypropyl]-2,4-dihydro-4-[4-[4-(4-Hydroxyphenyl)-1-piperazinyl]phenyl]-3H-1,24-triazol-3-one Antifungals(posaconazole etc)
5-Methoxy-2-[((4-methoxy-3,5-dimethyl-2-
 pyridinyl) methyl) thio]-1H-benzimidazole
 Antiulceratives (Omeprazole etc.)
2-Chloromethyl-3-methyl-4-(2,2,2-trifluoroethoxy) pyridine hydrochloride Antiulceratives (Lansoprazole etc.)
3-Methyl-4-[((2,2,2-trifluoro ethoxy-2-pyridinyl)methyl)thio]-1H-Benzimidazole Antiulceratives (Lansoprazole etc.)
Vanadyl Acetyl acetonate Antiulceratives (Lansoprazole etc.)
2-Chloromethyl-3,4-Dimethoxy Pyridine hydrochloride Antiulceratives (Pantoprazole Sodium etc)
5-Difluoromethoxy-2-Mercapto Benzimidazole Antiulceratives (Pantporazole Sodium etc)
5-Difluoromethoxy-2-[[(3,4-Dimethoxy-2-Pyridinyl) Methyl]-Thio]-1H-Benzimidazole Antiulceratives (Pantoprazole Sodium etc)
2,3-Dimethyl-4-Nitro Pyridine-1-Oxide Antiulceratives (Lansoprazole, Rabeprazole Sodium etc)
2-Hydroxymethyl-4-(3-MethoxyPropoxy)-3-Methyl Pyridine Hydrochloride Antiulceratives (Rabeprazole Sodium etc)
2-Chloromethyl-4-(3-MethoxyPropoxy)-3-Methyl Pyridine Hydrochloride Antiulceratives (Rabeprazole Sodium etc)
2-[[[4-(3-Methoxy Propoxy)-3-Methyl-2-Pyridinyl]Methyl] Thio]-1H-Benzimidazole Antiulceratives (Rabeprazole Sodium etc)
4-Chloro-2-Chloromethyl-3-methyl pyridine Hydrochloride Antiulceratives (Lansoprazole, Rabeprazole Sodium etc.)
4-Chloro-2,3-Dimethyl Pyridine-1-Oxide Hydrochloride Antiulceratives (Rabeprazole Sodium etc.)
2-[(4-Choloro-3-methyl-2-pyridinyl methyl)thio]-1H-benzimidazole Antiulceratives (Lansoprazole, Rabeprazole Sodium etc.)
2-[(3-Methyl-4-Nitro-2-pyridinyl methyl)thio]-1H-Benzimidazole Antiulceratives (Lansoprazole, Rabeprazole Sodium etc.)
Diethyl D(-) Tartrate Antiulceratives (ESOmeprazole Magnesium etc)
Cis-[2-Bromomethyl-2-(2,4-dichlorophenyl)-1,3-dioxolan-4-yl methyl] benzoate Antifungals (Itraconazole etc)
Cis-2-(2,4,-Dichlorophenyl)-2-(1H-1,2,4-triazol-1-yl methyl)-1,3-dioxolan-4-methanol methane sulfonate Antifungals (Itraconazole etc)
1-(4-Amino Phenyl)-4-(4-Methoxy Phenyl)Piperazine Antifungals (Itraconazole etc)
1-(4-Nitro Phenyl)-4-(4-Methoxy Phenyl)Piperazine Antifungals (Itraconazole etc)
2,4-Dihydro-4-[4-[(4-methoxy phenyl )-1-piperazinyl] phenyl]-2-(1- methylpropyl)-3H-1,2,4-trizol-3-one Antifungals (Itraconazole etc)
2,4-Dihydro-4-[4-[(4-Hydroxy phenyl )-1-piperazinyl] phenyl]-2-(1- methylpropyl)-3H-1,2,4-trizol-3-one Antifungals (Itraconazole etc)
Formamidine Acetate Antifungals (Itraconazole etc)
4-(4-Methoxyphenyl)-1-(1-methylethyl)piperazine Antifungals (Terconazole etc)
4-(4-Hydroxyphenyl)-1-(1-methylethyl)piperazine Antifungals (Terconazole etc)
1-(4-Chlorophenyl)Cyclobutane Carbonitrile Antiobesity(Sibutramine HCl etc.)
1-(4-Chlorophenyl)-1-(1-oxo-3-methylbutyl)cyclobutine Antiobesity(Sibutramine HCl etc.)
1-(4-Chlorophenyl)-α-(2-Methyl propyl) Cyclobutane Methanamine Hydrochloride Antiobesity(Sibutramine HCl etc.)
1-(4-Chlorophenyl)-N,N-dimethylpropyl) cyclobutane methanamine fumarate Antiobesity(Sibutramine HCl etc.)
1-(4-Chlorophenyl)-N-Formyl-α-(2-Methylpropyl)Cyclobutane Methanamine(subutramine Base) Antiobesity(Sibutramine HCl etc.)
1-(4-Chlorophenyl)-α-(2-Methyl propyl) Cyclobutane Methanamine Fumarate Antiobesity(Sibutramine HCl etc.)
2-Amino-3-cyano-5-Methyl Thiophene Antipsychotics(Olanapine etc.)
1-[(2,3-Dichlorophenyl) piperozine hydrochloride Antipsychotics(Aripiprazole etc) 83
2-(2-Nitro aniline)-s-Methyl Thiophene-3- Carbonitrile Antipsychotics(Olanapine etc.)
2-Methyl-4-amino-10H-thieno-[2,3-b ] [1,5] Benzodiazepine Hydrochloride Antipsychotics(Olanapine etc.)
2-Methyl-4-(1-piperazinyl)-10H-Thieno[2,3-b][1,5]Benzodiazepine Antipsychotics(Olanapine etc.)
Dibenzo-[b,f][1,4]Thiazepin-11(10H)-One] Antipsychotics(Quetiapine Hemifumarate etc.)
2-(2-Nitro anilino)-5-methyl thiophene-3-carbonitrile Antipsychotics(Olanapine etc.)
N-[Dibenzo-[b,f][1,4]Thiazepin-11-Yl]Piperrazine Dihydrochloride Antipsychotics(Quetiapine Hemifumarate etc.)
2-[2-(1-Piperazintl) ethoxy] ethanol Antipsychotics (Quetiapine Hemifumarate etc.)
2-[2-(1-Piperazinyl) ethoxy] ethanol DiHydrochloride Antipsychotics (Quetiopine Hemifumarate etc.)
10-Hydroxy-8-Chlorodibenzo[b,f]thiepine Antipsychotics(Zotepine etc.)
7-Hydroxy-3,4-Dihydro-2(1H)-Quinolinone) Antipsychotics(Aripiprazole etc.)
1-(2,3-Dichlorophenyl) Piperazine) Antipsychotics(Aripiprazole etc.)
(S)-(-)-3-(Dimethyl amino)-1-(2-Thienyl)-1-Propanol Antidepressants(Duloxetine HCL etc.)
N,N-Dimethyl-3-(1-Naphthalenylaxy)-3-(2-Thienyl)-1- propanamine oxalate Antidepressants (Duloxetine HCL etc.)
5-[(2R)-2-Amino Propyl]-2-Methoxy Benzene Sulfonamide Treatment of BPH (Tamsulosin HCL etc.)
4-Hydrazino-N-Methyl Benzene Methane Sulfonamide HCL Antimigraines (Sumatriptan etc)
4-Chloro butyraldehyde Sodium Bisulphite Adduct Antimigraines (Sumatriptan etc)
4-(Pyrrolidino Sulfonyl Methyl) Phenylhydrazine Hydrochloride Monohydrate Antimigraines(Almotriptan Malate etc.)
4-(Pyrrolidino Sulfonyl Methyl) Nitrobenzene Antimigraines(Almotriptan Malate etc.)
4-((1H-1,2,4-triazol-1-yl)methyl) benzeneamine Antimigraines(Rizatriptan Benzoate etc.)
1-(4-Nitrobenzyl)-1H-1,2,4-triazole Antimigranies(Rizatriptan Benzoate etc.)
(4S)-4-(4-Aminobenzyl)-2-oxazolidinone Antimigraines(Zolmitriptan etc.)
4-Dimethylamino butyraldehydediethyl acetal Antimigraines(Zolmitriptan, Rizatriptan etc.)
5-α,α,α',α'-Pentamethyl-1,3-benzenediacetonitrile Antineoplastics(Anastrozole etc.)
2,2'-(5-Bromomethyl-1,3-phenylene)di(2-methylpropionitrile) Antineoplastics(Anastrozole etc.)
N-(5-Bromo-2-methyl phenyl)-4-(3-pyrudyl)-2-pyrimidineamine Antineoplastics(Imatinib Mesylate etc.)
6-Methyl-N'-4-(Pyridin-3-yl)Pyrimidin-2-yl)benzene-1,3-diamine Antineoplastics(Imatinib methane sulfonate etc.)
4-((4-Methylpiperazinyl-1-yl)methyl)benzoic acid dihydrochloride Antineoplastics (Imatinib methane sulfonate etc.
(S)-(-)-2,6-Diamino-4,5,6,7-tetrahydro Benzothiazole Antiparkinsonians(Pramipexole Dihydrochloride etc.)
(+)-2,6-Diamino-4,5,6,7-tetrahydro Benzothiazole Antiparkinsonians(Pramipexole Dihydrochloride etc.)
4-Acrtamido Cyclohexanone Antiparkinsonians(Pramipexole Dihydrochloride etc.)
5-Benzoyl-7-Bromo-2,3-Dihydro-1H-Pyrrolizine-1-Carboxylic Acid Analgesic, Anti-inflammatory(Ketorolac Tromethamine etc.)
(S,S)-2,8-Diazabicyclo[4.3.0]nonane Antibacterials(moxifloxacin HCl etc.)
3-[(2-Hydroxy)-1-ethyl]-5-[N-methyl(methanesulfonamide)]-1H-indole-2-Carboxylicacid methyl ester Antimigraines(Sumatripton Succinate etc.)
[3-(2-Aminoethyl)-1H-indol-5-yl]-N-methyl methane sulfonamide Antimigraines(Sumatriptan Succinate etc.)
3-[2-Dimethylamino)ethyl]-N-methyl-1H-indole-5-methane sulfonamide(Sumatriptan Base) Antimigraines(Sumatriptan Succinate etc)
α-α-Diphenyl-4-piperazine methanol(Azacyclonol) Antihistaminics(Fexofenadine HCl etc.)
2-(4-{4-[4-(Hydroxy-diphnyl-methyl)-piperidin-1-yl]butanoyl}phenyl)-2-methyl-propionic acid Antihistaminics(Fexofenadine HCl etc)
((4-(4-Fluorophenyl)-6-isopropyl-2-(N-methyl-N-Methylsulfonamido)pyrimidin-5-yl)methyl)trimethylphosphonium bromide Antilipemics(rosuvastatin SCalcium etc.)